摘要：【中文】本发明涉及一种伊马替尼及其甲磺酸盐的合成方法，其包括以下步骤：以3‑乙酰吡啶和N,N‑二甲基酰胺二甲基缩醛为起始原料经缩合得到3‑二甲氨基‑1‑(3‑吡啶基)‑2‑丙烯‑1‑酮，再和2‑甲基‑5‑硝基苯基胍硝酸盐成嘧啶环，经硝基还原得到N‑(5‑氨基‑2‑甲基苯基)‑4‑(3‑吡啶基)‑2‑嘧啶胺，和对氯甲基苯甲酰氯酰胺化，再和1‑甲基哌嗪亲和取代得到伊马替尼，最后和甲磺酸成盐。本发明的方法得到的产品杂质少，后处理简单，总收率高，绿色环保安全，适合大规模工业化生产甲磺酸伊马替尼生产工艺。 【EN】The invention relates to a method for synthesizing imatinib and mesylate thereof, which comprises the following steps: the method comprises the steps of condensing 3-acetylpyridine and N, N-dimethyl amide dimethyl acetal serving as starting materials to obtain 3-dimethylamino-1- (3-pyridyl) -2-propen-1-one, forming a pyrimidine ring with 2-methyl-5-nitrophenylguanidine nitrate, reducing the pyrimidine ring through nitro to obtain N- (5-amino-2-methylphenyl) -4- (3-pyridyl) -2-pyrimidinamine, amidating p-chloromethyl benzoyl chloride, carrying out affinity substitution with 1-methylpiperazine to obtain imatinib, and finally salifying with methanesulfonic acid. The product obtained by the method has the advantages of less impurities, simple post-treatment, high total yield, environmental protection and safety, and is suitable for large-scale industrial production of imatinib mesylate.

摘要：【中文】本发明涉及通式(I)化合物或其异构体、其水合物或其药学上可接受的盐。本发明还涉及所述化合物或其异构体、其水合物或其药学上可接受的盐的制备方法、含有其的药用组合物及其在制备药物中的用途，所述药物用于抗血小板聚集和治疗相关疾病例如抗血栓。 【EN】The invention relates to a compound of a general formula (I) or an isomer, a hydrate or a pharmaceutically acceptable salt thereof. The invention also relates to a preparation method of the compound or the isomer thereof, the hydrate thereof or the pharmaceutically acceptable salt thereof, a medicinal composition containing the compound and application thereof in preparing medicaments for resisting platelet aggregation and treating related diseases such as thrombosis.

摘要：【中文】本申请提供一种报文处理方法及装置，涉及通信领域。本申请通过获取数据报文的IPv6地址、以及IPv6地址对应的用户角色，将IPv6地址与用户角色进行映射，生成IPv6地址的映射标识，根据映射标识，按照访问控制列表ACL的匹配策略对数据报文进行转发，可以减少按照ACL列表执行ACL策略时所占用的交换机硬件资源。 【EN】The application provides a message processing method and device, and relates to the field of communication. The method and the device have the advantages that the IPv6 address of the data message and the user role corresponding to the IPv6 address are obtained, the IPv6 address and the user role are mapped, the mapping identifier of the IPv6 address is generated, the data message is forwarded according to the mapping identifier and the matching strategy of the access control list ACL, and occupied switch hardware resources can be reduced when the ACL strategy is executed according to the ACL list.

摘要：【中文】本发明公开了一种侵彻过载信号的特征提取方法，包括利用总体经验模态分解法对测试信号进行分解、构造多维观察信号并对多维观察信号的自相关矩阵进行奇异值分解、确定主分量信号源数、形成多通道混合信号、采用二阶盲辨识算法对多通道混合信号进行盲源分离处理获得源信号、对源信号进行特征提取；针对合理分离弹体侵彻板靶时弹体的刚体加速度特征，滤除测试信号中含有的结构响应和外部噪声成份，从而进行侵彻过载信号特征的提取的问题，本发明所提供的一种侵彻过载信号的特征提取方法，对侵彻过载信号进行处理，能够获得反映弹体侵彻目标过程的刚体加速度特征的信号分量及弹体侵彻目标过程时的弹体二次或多次谐振频率的信号分量。 【EN】The invention discloses a characteristic extraction method of penetration overload signals, which comprises the steps of decomposing test signals by using a general empirical mode decomposition method, constructing multi-dimensional observation signals, carrying out singular value decomposition on an autocorrelation matrix of the multi-dimensional observation signals, determining the number of principal component signal sources, forming multi-channel mixed signals, carrying out blind source separation processing on the multi-channel mixed signals by adopting a second-order blind identification algorithm to obtain source signals, and carrying out characteristic extraction on the source signals; aiming at reasonably separating rigid acceleration characteristics of a projectile body when the projectile body penetrates a plate target and filtering structural response and external noise components contained in a test signal so as to extract penetration overload signal characteristics, the method for extracting penetration overload signal characteristics provided by the invention is used for processing penetration overload signals and can obtain signal components reflecting rigid acceleration characteristics of the projectile body in a penetration target process and signal components of secondary or multiple resonance frequencies of the projectile body in the penetration target process.

摘要：【中文】本发明提供了一种用于车载导航的信息处理方法，包括：获取收藏地址及相关联的收藏地址标识，所述收藏地址标识包括表征所述收藏地址的标识字段；将所述收藏地址与所述收藏地址标识相关联地存储于导航通讯录中；获取导航指令；从所述导航指令提取目的地标识，所述目的地标识包括表征导航目的地的标识字段；对所述目的地标识执行扩展，以获得扩展目的地标识，所述扩展目的地标识的至少一个标识字段被扩展为对应的同义词组；基于所述扩展目的地标识查找所述导航通讯录以确定所述导航目的地；以及基于所述导航目的地规划导航路线。 【EN】The invention provides an information processing method for vehicle navigation, which comprises the following steps: acquiring a collection address and a relevant collection address identifier, wherein the collection address identifier comprises an identifier field for representing the collection address; storing the collection address and the collection address identification in a navigation address book in a correlated manner; acquiring a navigation instruction; extracting a destination identification from the navigation instruction, the destination identification including an identification field characterizing a navigation destination; performing expansion on the destination identifier to obtain an expanded destination identifier, wherein at least one identification field of the expanded destination identifier is expanded into a corresponding synonym group; searching the navigation address book based on the extended destination identifier to determine the navigation destination; and planning a navigation route based on the navigation destination.

摘要：【中文】本发明提供一种报文转发控制方法及装置，所述方法包括：获取本交换机接入的第一终端设备以及远端汇聚交换机接入的第二终端设备的安全组标签SGT，并维护第一终端设备的IP地址与SGT的对应关系，以及第二终端设备的IP地址与SGT的对应关系；当从终端侧接收到第一报文时，分别基于所述第一报文的源IP地址以及目的IP地址，查询所述第一终端设备的IP地址与SGT的对应关系，以及第二终端设备的IP地址与SGT的对应关系，以确定第一源SGT以及第一目的SGT；基于所述第一源SGT以及第一目的SGT对所述第一报文进行转发控制。应用本发明实施例可以减少源网关和目的网关之间的网络带宽的浪费，并减少网络安全隐患。 【EN】The invention provides a message forwarding control method and a device, wherein the method comprises the following steps: acquiring security group labels SGT of a first terminal device accessed by the switch and a second terminal device accessed by a remote convergence switch, and maintaining the corresponding relation between the IP address of the first terminal device and the SGT and the corresponding relation between the IP address of the second terminal device and the SGT; when a first message is received from a terminal side, respectively inquiring the corresponding relation between the IP address of the first terminal equipment and the SGT and the corresponding relation between the IP address of the second terminal equipment and the SGT based on the source IP address and the destination IP address of the first message so as to determine a first source SGT and a first destination SGT; and performing forwarding control on the first message based on the first source SGT and the first destination SGT. By applying the embodiment of the invention, the waste of network bandwidth between the source gateway and the destination gateway can be reduced, and the potential safety hazard of the network can be reduced.

摘要：【中文】本申请提供了业务访问方法和装置。本申请中，当第一主机对第二主机进行业务访问时，不再要求第一主机发送的业务访问报文中携带第一主机匹配的第一用户角色，而是由第一主机的边缘设备即源Border依据业务访问报文的源IP地址确定第一主机匹配的第一用户角色以及依据业务访问报文的目的IP地址确定第二主机匹配的第二用户角色，并且源Border还对第一主机的业务访问进行策略控制，以在第一主机不具有访问第二主机的权限时，在源Border端就可禁止业务访问报文转发。本申请能够实现在业务访问报文中不携带用户角色的前提下实现业务访问，且由源Border对第一主机的业务访问进行策略控制，减少网络负载。 【EN】The application provides a service access method and device. In the application, when a first host accesses a second host, a service access message sent by the first host is no longer required to carry a first user role matched with the first host, but an edge device of the first host, namely, a source Border, determines a first user role matched with the first host according to a source IP address of the service access message and a second user role matched with the second host according to a destination IP address of the service access message, and the source Border also performs policy control on service access of the first host, so that when the first host does not have the authority of accessing the second host, forwarding of the service access message can be prohibited at a source Border end. According to the method and the device, the service access can be realized on the premise that the service access message does not carry the user role, the strategy control is carried out on the service access of the first host by the source Border, and the network load is reduced.

摘要：【中文】本发明公开了一种冲击信号特征提取及降噪方法，包括步骤利用相空间重构理论重构吸引子轨迹矩阵、对子矩阵B进行奇异值分解、确定重构子矩阵B的最佳行数、确定重构子矩阵B的有效阶次和重构子矩阵B，获得降噪后的冲击信号；针对现有技术中小波消噪方法存在降噪处理效果不理想，降噪后的冲击信号信噪比低的问题，本发明所提供的一种冲击信号特征提取及降噪方法，降噪处理效果理想,降噪处理后重构的信号具有较高的信噪比。 【EN】The invention discloses an impact signal characteristic extraction and noise reduction method, which comprises the steps of reconstructing an attractor track matrix by utilizing a phase space reconstruction theory, carrying out singular value decomposition on a submatrix B, determining the optimal row number of the reconstructed submatrix B, determining the effective order of the reconstructed submatrix B and reconstructing the submatrix B, and obtaining an impact signal subjected to noise reduction; aiming at the problems that the wavelet denoising method in the prior art is not ideal in denoising effect and the signal-to-noise ratio of denoised impulse signals is low, the impulse signal feature extraction and denoising method provided by the invention is ideal in denoising effect, and reconstructed signals after denoising have higher signal-to-noise ratio.

摘要：【中文】本申请涉及神经网络技术领域，尤其涉及一种神经网络模型训练方法、分类方法、装置和电子设备。其中，神经网络模型训练方法包括：获取当前应用场景对应的神经网络初始模型和当前应用场景对应的实际样本集；该神经网络初始模型的至少一个网络层包含有多个激活函数；通过实际样本集训练所述神经网络初始模型，以从至少一个网络层包含的多个激活函数中确定最优激活函数；将确定出最优激活函数的神经网络初始模型，作为当前应用场景的神经网络模型。相比激活函数单一且固定的模型，本申请训练的模型具有较好的通用性和扩展性，提升了模型的训练灵活性和效率。 【EN】The present application relates to the field of neural network technologies, and in particular, to a neural network model training method, a neural network model classification device, and an electronic device. The neural network model training method comprises the following steps: acquiring a neural network initial model corresponding to a current application scene and an actual sample set corresponding to the current application scene; at least one network layer of the initial neural network model comprises a plurality of activation functions; training the neural network initial model through an actual sample set to determine an optimal activation function from a plurality of activation functions contained in at least one network layer; and taking the neural network initial model of the determined optimal activation function as the neural network model of the current application scene. Compared with a model with a single and fixed activation function, the model trained by the method has better universality and expansibility, and the training flexibility and efficiency of the model are improved.

摘要：【中文】本发明公开了一种高速垂直循环停车设备，包括一套后框架、一套防摆组件、两套提升链条、一套提升系统，一套前框架、两套底部导向轮组、至少四套载车板，整体通过后框架和前框架的四个立柱安装于地面基础上，提升系统的大驱动轮和提升链条的带轴承滚轮通过啮合运动来实行旋转提升，防摆轨道整体上下对称、左右对称、接近封闭的结构保证运行过程中始终有两个主导向轮和防摆轨道严格支撑。本发明停车设备主要用于地面停车场改造立体车位，尤其是适合建设高层垂直循环停车设备，可实现提升速度的成倍增加以减少设备存取车运行时间，改进的防摆结构保证载车板运行过程安全可靠，提高了该类型停车设备使用的便捷性。 【EN】The invention discloses high-speed vertical circulation parking equipment which comprises a set of rear frame, a set of anti-swing assembly, two sets of lifting chains, a set of lifting system, a set of front frame, two sets of bottom guide wheel sets and at least four sets of vehicle carrying plates. The parking equipment is mainly used for transforming the three-dimensional parking spaces in ground parking lots, is particularly suitable for building high-rise vertical circulation parking equipment, can realize the multiplied increase of the lifting speed so as to reduce the operation time of equipment for storing and taking vehicles, and the improved anti-swing structure ensures the safe and reliable operation process of the vehicle carrying plate and improves the use convenience of the parking equipment of the type.